G007-LK
Descripción del producto
Name | 4-[5-[(1E)-2-[4-(2-Chlorophenyl)-5-[5-(methylsulfonyl)-2-pyridinyl]-4H-1,2,4-triazol-3-yl]ethenyl]-1,3,4-oxadiazol-2-yl]benzonitrile | |
Molecular Structure | ||
Molecular Formula | C25H16ClN7O3S | |
Molecular Weight | 529.96 | |
CAS Registry Number | 1380672-07-0 |
G007-LK displays high selectivity toward tankyrases 1 and 2 with biochemical IC50 values of 46 nM and 25 nM, respectively, and a cellular IC50 value of 50 nM combined with an excellent pharmacokinetic profile in mice. |
Grupos de Producto : Síntesis personalizada
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